TargetMol

Olorinab

Product Code:
 
TAR-T14302
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14302-1mg1mg£111.00
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TAR-T14302-5mg5mg£168.00
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TAR-T14302-10mg10mg£229.00
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TAR-T14302-25mg25mg£389.00
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TAR-T14302-50mg50mg£544.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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  • Further Information
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Further Information

Bioactivity:
Olorinab (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.
CAS:
1268881-20-4
Formula:
C18H23N5O3
Molecular Weight:
357.414
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
[H][C@@]12C[C@]1([H])c1c(C2)c(nn1-c1cn(=O)ccn1)C(=O)N[C@H](CO)C(C)(C)C
Target:
Cannabinoid Receptor

Documents

References

Han S, et al. Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain. ACS Med Chem Lett. 2017 Nov 30;8(12):1309-1313.