TargetMol

PROTAC ERRα Degrader-2

Product Code:
 
TAR-T18609
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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Further Information

Bioactivity:
PROTAC ERRα Degrader-2 is a compound consisting of an MDM2 ligand binding group, a linker, and an estrogen-related receptor alpha (ERRα) binding group. This compound is designed to specifically degrade estrogen-related receptor alpha (ERRα), acting as an ERRα degrader[1].
CAS:
2306388-85-0
Molecular Weight:
1150.99
Purity:
0.98
SMILES:
C(=O)(N1[C@]([C@](N=C1C2=C(OC(C)C)C=C(OC)C=C2)(C3=CC=C(Cl)C=C3)[H])(C4=CC=C(Cl)C=C4)[H])N5CC(=O)N(CC(NCCCCCNC(/C(=C/C6=CC(OC)=C(OCC7=C(C(F)(F)F)C=C(C(F)(F)F)C=C7)C=C6)/C#N)=O)=O)CC5

Documents

References

Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor ? (ERR?) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772.